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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T72188 | Nicotinamide Hydrochloride | Niacinamide Hydrochloride,Nicotinic acid amide Hydrochloride,Niacinamide Hydrochloride ; Nicotinic acid amide Hydrochloride | |
Nicotinamide Hydrochloride is a form of vitamin B3 or niacin that inhibits sirtuin 2 ( SIRT2 ) activity in vitro , with an EC 50 of 2 μM. Nicotinamide Hydrochloride inhibits up to 90% melanoma cell number and increases c... | |||
T33666 | Nicotinamide, N-(m-difluoromethoxyphenyl)-, hydrochloride | ||
Nicotinamide, N-(m-difluoromethoxyphenyl)-, hydrochloride is a bioactive chemical. | |||
T4853 | TRIA-662 | 3-Carbamoyl-1-methylpyridinium Chloride,1-Methylnicotinamide chloride,1-methylpyridin-1-ium-3-carboxamide hydrochloride,Nicotinamide Chloromethylate | Others , Endogenous Metabolite |
TRIA-662 (Nicotinamide Chloromethylate) is a niacin metabolite excreted via the urinary system. | |||
T40855 | LB-60-OF61 hydrochloride | LB-60-OF61 hydrochloride | |
LB-60-OF61 hydrochloride is a highly effective inhibitor of NAMPT, a key enzyme involved in the transfer of nicotinamide phosphoribosyl groups. This compound, known for its cytotoxic properties, specifically targets cell... | |||
T22785 | FK 866 hydrochloride (658084-64-1 free base) | FK 866 hydrochloride | Others |
FK 866 hydrochloride is an inhibitor of nicotinamide phosphoribosyltransferase (IC50: 0.09nM and 27.2nM). | |||
T22801 | GNE-617 hydrochloride (1362154-70-8 free base) | GNE-617 hydrochloride | Others |
GNE-617 hydrochloride is a potent and competitive inhibitor of nicotinamide phosphoribosyltransferase (IC50: 5nM). GNE-617 hydrochloride reduces the NAD levels in a > 95% reduction in both NAPRT1-deficient and NAPRT1-pro... | |||
T37578 | GPP 78 hydrochloride | ||
GPP 78 hydrochloride is a potent inhibitor of nicotinamide phosphoribosyltransferase (Nampt) with an IC50 of 3 nM for NAD depletion. GPP 78 hydrochloride is toxic to neuroblastoma cells SH-SY5Y via induction of autophagy... | |||
T78164 | JBSNF-000028 hydrochloride | Others | |
JBSNF-000028 hydrochloride is a potent inhibitor of nicotinamide N-methyltransferase (NNMT) with IC50 values of 0.033 μM for human NNMT (hNNMT), 0.19 μM for monkey NNMT (mkNNMT), and 0.21 μM for mouse NNMT (mNNMT). This ... |